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PDB: 1 results

6KYA
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BU of 6kya by Molmil
Crystal structure of human TLR8 in complex TH1027
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 3-[5-methylsulfanyl-4-(3,4,5-trimethylphenyl)-1,2,4-triazol-3-yl]propan-1-ol, ...
Authors:Tanji, H, Sakaniwa, K, Ohto, U, Shimizu, T.
Deposit date:2019-09-17
Release date:2020-05-27
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (2.89 Å)
Cite:Rationally Designed Small-Molecule Inhibitors Targeting an Unconventional Pocket on the TLR8 Protein-Protein Interface.
J.Med.Chem., 63, 2020

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