5RXN
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![BU of 5rxn by Molmil](/molmil-images/mine/5rxn) | |
4RXN
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![BU of 4rxn by Molmil](/molmil-images/mine/4rxn) | |
7UPJ
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![BU of 7upj by Molmil](/molmil-images/mine/7upj) | HIV-1 PROTEASE/U101935 COMPLEX | Descriptor: | HIV-1 PROTEASE, N-(3-CYCLOPROPYL(5,6,7,8,9,10-HEXAHYDRO-2-OXO-2H-CYCLOOCTA[B]PYRAN-3-YL)METHYL)PHENYLBENZENSULFONAMIDE | Authors: | Watenpaugh, K.D, Janakiraman, M.N. | Deposit date: | 1996-12-05 | Release date: | 1997-04-21 | Last modified: | 2024-04-03 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Structure-based design of nonpeptidic HIV protease inhibitors: the sulfonamide-substituted cyclooctylpyramones. J.Med.Chem., 40, 1997
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1FX1
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![BU of 1fx1 by Molmil](/molmil-images/mine/1fx1) | |
5UPJ
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![BU of 5upj by Molmil](/molmil-images/mine/5upj) | HIV-2 PROTEASE/U99283 COMPLEX | Descriptor: | 5,6,7,8,9,10-HEXAHYDRO-4-HYDROXY-3-(1-PHENYLPROPYL)CYCLOOCTA[B]PYRAN-2-ONE, HIV-2 PROTEASE | Authors: | Watenpaugh, K.D, Mulichak, A.M, Finzel, B.C. | Deposit date: | 1996-12-10 | Release date: | 1997-04-21 | Last modified: | 2024-04-03 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Use of medium-sized cycloalkyl rings to enhance secondary binding: discovery of a new class of human immunodeficiency virus (HIV) protease inhibitors. J.Med.Chem., 38, 1995
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6UPJ
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![BU of 6upj by Molmil](/molmil-images/mine/6upj) | HIV-2 PROTEASE/U99294 COMPLEX | Descriptor: | 6,7,8,9-TETRAHYDRO-4-HYDROXY-3-(1-PHENYLPROPYL)CYCLOHEPTA[B]PYRAN-2-ONE, HIV-2 PROTEASE | Authors: | Watenpaugh, K.D, Mulichak, A.M, Finzel, B.C. | Deposit date: | 1996-12-10 | Release date: | 1997-04-21 | Last modified: | 2024-04-03 | Method: | X-RAY DIFFRACTION (2.34 Å) | Cite: | Use of medium-sized cycloalkyl rings to enhance secondary binding: discovery of a new class of human immunodeficiency virus (HIV) protease inhibitors. J.Med.Chem., 38, 1995
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1HPO
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![BU of 1hpo by Molmil](/molmil-images/mine/1hpo) | HIV-1 PROTEASE TRIPLE MUTANT/U103265 COMPLEX | Descriptor: | 4-CYANO-N-(3-CYCLOPROPYL(5,6,7,8,9,10-HEXAHYDRO-4-HYDROXY-2-OXO-CYCLOOCTA[B]PYRAN-3-YL)METHYL)PHENYL BENZENSULFONAMIDE, HIV-1 PROTEASE | Authors: | Watenpaugh, K.D, Janakiraman, M.N. | Deposit date: | 1996-12-10 | Release date: | 1997-04-21 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Structure-based design of nonpeptidic HIV protease inhibitors: the sulfonamide-substituted cyclooctylpyramones. J.Med.Chem., 40, 1997
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2UPJ
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![BU of 2upj by Molmil](/molmil-images/mine/2upj) | |
3UPJ
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![BU of 3upj by Molmil](/molmil-images/mine/3upj) | |
4UPJ
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![BU of 4upj by Molmil](/molmil-images/mine/4upj) | |
1UPJ
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1QB0
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![BU of 1qb0 by Molmil](/molmil-images/mine/1qb0) | HUMAN CDC25B CATALYTIC DOMAIN | Descriptor: | BETA-MERCAPTOETHANOL, CHLORIDE ION, PROTEIN (M-PHASE INDUCER PHOSPHATASE 2 (CDC25B)), ... | Authors: | Watenpaugh, K.D, Reynolds, R.A. | Deposit date: | 1999-04-29 | Release date: | 2000-04-29 | Last modified: | 2018-02-28 | Method: | X-RAY DIFFRACTION (1.91 Å) | Cite: | Crystal structure of the catalytic subunit of Cdc25B required for G2/M phase transition of the cell cycle. J.Mol.Biol., 293, 1999
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1JSV
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![BU of 1jsv by Molmil](/molmil-images/mine/1jsv) | |
1CWT
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![BU of 1cwt by Molmil](/molmil-images/mine/1cwt) | HUMAN CDC25B CATALYTIC DOMAIN WITH METHYL MERCURY | Descriptor: | CDC25 B-TYPE TYROSINE PHOSPHATASE, CHLORIDE ION, METHYL MERCURY ION, ... | Authors: | Watenpaugh, K.D, Reynolds, R.A. | Deposit date: | 1999-08-26 | Release date: | 2000-08-30 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Crystal structure of the catalytic subunit of Cdc25B required for G2/M phase transition of the cell cycle. J.Mol.Biol., 293, 1999
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1D4S
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![BU of 1d4s by Molmil](/molmil-images/mine/1d4s) | HIV-1 PROTEASE V82F/I84V DOUBLE MUTANT/TIPRANAVIR COMPLEX | Descriptor: | N-(3-{(1R)-1-[(6R)-4-HYDROXY-2-OXO-6-PHENETHYL-6-PROPYL-5,6-DIHYDRO-2H-PYRAN-3-YL]PROPYL}PHENYL)-5-(TRIFLUOROMETHYL)-2-PYRIDINESULFONAMIDE, PROTEIN (HIV-1 PROTEASE) | Authors: | Watenpaugh, K.D, Janakiraman, M.N. | Deposit date: | 1999-10-05 | Release date: | 1999-10-12 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Structure-based design of HIV protease inhibitors: sulfonamide-containing 5,6-dihydro-4-hydroxy-2-pyrones as non-peptidic inhibitors. J.Med.Chem., 39, 1996
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1CWR
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![BU of 1cwr by Molmil](/molmil-images/mine/1cwr) | |
1CWS
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![BU of 1cws by Molmil](/molmil-images/mine/1cws) | HUMAN CDC25B CATALYTIC DOMAIN WITH TUNGSTATE | Descriptor: | BETA-MERCAPTOETHANOL, CDC25 B-TYPE TYROSINE PHOSPHATASE, CHLORIDE ION, ... | Authors: | Watenpaugh, K.D, Reynolds, R.A, Chidester, C.G. | Deposit date: | 1999-08-26 | Release date: | 2000-08-30 | Last modified: | 2011-07-13 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Crystal structure of the catalytic subunit of Cdc25B required for G2/M phase transition of the cell cycle. J.Mol.Biol., 293, 1999
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1D4Y
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![BU of 1d4y by Molmil](/molmil-images/mine/1d4y) | HIV-1 PROTEASE TRIPLE MUTANT/TIPRANAVIR COMPLEX | Descriptor: | N-(3-{(1R)-1-[(6R)-4-HYDROXY-2-OXO-6-PHENETHYL-6-PROPYL-5,6-DIHYDRO-2H-PYRAN-3-YL]PROPYL}PHENYL)-5-(TRIFLUOROMETHYL)-2-PYRIDINESULFONAMIDE, PROTEIN (HIV-1 PROTEASE) | Authors: | Watenpaugh, K.D, Janakiraman, M.N. | Deposit date: | 1999-10-06 | Release date: | 1999-10-13 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (1.97 Å) | Cite: | Structure-based design of HIV protease inhibitors: sulfonamide-containing 5,6-dihydro-4-hydroxy-2-pyrones as non-peptidic inhibitors. J.Med.Chem., 39, 1996
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5FX2
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![BU of 5fx2 by Molmil](/molmil-images/mine/5fx2) | |
2FX2
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![BU of 2fx2 by Molmil](/molmil-images/mine/2fx2) | |
4FX2
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![BU of 4fx2 by Molmil](/molmil-images/mine/4fx2) | |
3FX2
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![BU of 3fx2 by Molmil](/molmil-images/mine/3fx2) | |
1F4P
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![BU of 1f4p by Molmil](/molmil-images/mine/1f4p) | Y98W FLAVODOXIN MUTANT 1.5A (D. VULGARIS) | Descriptor: | FLAVIN MONONUCLEOTIDE, FLAVODOXIN | Authors: | Reynolds, R.A, Watt, W, Watenpaugh, K.D. | Deposit date: | 2000-06-08 | Release date: | 2001-04-04 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (1.3 Å) | Cite: | Structures and comparison of the Y98H (2.0 A) and Y98W (1.5 A) mutants of flavodoxin (Desulfovibrio vulgaris). Acta Crystallogr.,Sect.D, 57, 2001
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2HPE
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2HPF
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![BU of 2hpf by Molmil](/molmil-images/mine/2hpf) | |