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PDB: 1 results

4L6Q
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BU of 4l6q by Molmil
ROCK2 in complex with benzoxaborole
Descriptor: 6-[4-(aminomethyl)-2-fluorophenoxy]-2,1-benzoxaborol-1(3H)-ol, Rho-associated protein kinase 2
Authors:Rock, F, Jarnagin, K.
Deposit date:2013-06-12
Release date:2013-10-02
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2.79 Å)
Cite:Linking phenotype to kinase: identification of a novel benzoxaborole hinge-binding motif for kinase inhibition and development of high-potency rho kinase inhibitors.
J.Pharmacol.Exp.Ther., 347, 2013

220113

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