4TRL
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![BU of 4trl by Molmil](/molmil-images/mine/4trl) | Structure of Ephrin type-A receptor 2 | Descriptor: | Ephrin type-A receptor 2 | Authors: | Wei, Q, Wang, N. | Deposit date: | 2014-06-17 | Release date: | 2014-07-02 | Last modified: | 2023-12-27 | Method: | X-RAY DIFFRACTION (2.452 Å) | Cite: | Structure of Ephrin type-A receptor 2 To Be Published
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5CIO
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![BU of 5cio by Molmil](/molmil-images/mine/5cio) | Crystal structure of PqqF | Descriptor: | ZINC ION, pyrroloquinoline quinone biosynthesis protein PqqF | Authors: | Wei, Q, Xu, D, Ran, T, Wang, W. | Deposit date: | 2015-07-13 | Release date: | 2016-06-08 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Crystal Structure and Function of PqqF Protein in the Pyrroloquinoline Quinone Biosynthetic Pathway J.Biol.Chem., 291, 2016
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5EK7
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![BU of 5ek7 by Molmil](/molmil-images/mine/5ek7) | |
6ITX
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![BU of 6itx by Molmil](/molmil-images/mine/6itx) | |
7VXO
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![BU of 7vxo by Molmil](/molmil-images/mine/7vxo) | |
7X5T
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![BU of 7x5t by Molmil](/molmil-images/mine/7x5t) | |
2R28
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![BU of 2r28 by Molmil](/molmil-images/mine/2r28) | |
2F2O
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![BU of 2f2o by Molmil](/molmil-images/mine/2f2o) | |
2F2P
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![BU of 2f2p by Molmil](/molmil-images/mine/2f2p) | |
4IL1
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![BU of 4il1 by Molmil](/molmil-images/mine/4il1) | Crystal Structure of the Rat Calcineurin | Descriptor: | CALCIUM ION, Calmodulin, Calcineurin subunit B type 1, ... | Authors: | Ye, Q, Faucher, F, Jia, Z. | Deposit date: | 2012-12-28 | Release date: | 2013-10-02 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (3 Å) | Cite: | Structural basis of calcineurin activation by calmodulin. Cell Signal, 25, 2013
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7U9Y
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![BU of 7u9y by Molmil](/molmil-images/mine/7u9y) | |
7UAS
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![BU of 7uas by Molmil](/molmil-images/mine/7uas) | |
8WD8
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![BU of 8wd8 by Molmil](/molmil-images/mine/8wd8) | Cryo-EM structure of TtdAgo-guide DNA-target DNA complex | Descriptor: | Argonaute family protein, Guide DNA, MAGNESIUM ION, ... | Authors: | Zhuang, L. | Deposit date: | 2023-09-14 | Release date: | 2024-01-31 | Last modified: | 2024-05-01 | Method: | ELECTRON MICROSCOPY (2.9 Å) | Cite: | Molecular mechanism for target recognition, dimerization, and activation of Pyrococcus furiosus Argonaute. Mol.Cell, 84, 2024
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8XJ3
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![BU of 8xj3 by Molmil](/molmil-images/mine/8xj3) | |
7JWI
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![BU of 7jwi by Molmil](/molmil-images/mine/7jwi) | |
7JWJ
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![BU of 7jwj by Molmil](/molmil-images/mine/7jwj) | Crystal Structure of B17-C1 TCR-H2Db | Descriptor: | B17.C1 TCR alpha chain, B17.C1 TCR beta chain, Beta-2-microglobulin, ... | Authors: | Farenc, C, Rossjohn, J, Gras, S, Szeto, C. | Deposit date: | 2020-08-25 | Release date: | 2021-07-07 | Last modified: | 2024-04-24 | Method: | X-RAY DIFFRACTION (3.251 Å) | Cite: | Canonical T cell receptor docking on peptide-MHC is essential for T cell signaling. Science, 372, 2021
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6J6M
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![BU of 6j6m by Molmil](/molmil-images/mine/6j6m) | Co-crystal structure of BTK kinase domain with Zanubrutinib | Descriptor: | (7S)-2-(4-phenoxyphenyl)-7-(1-propanoylpiperidin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide, IMIDAZOLE, Tyrosine-protein kinase BTK | Authors: | Zhou, X, Hong, Y. | Deposit date: | 2019-01-15 | Release date: | 2019-10-23 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (1.25 Å) | Cite: | Discovery of Zanubrutinib (BGB-3111), a Novel, Potent, and Selective Covalent Inhibitor of Bruton's Tyrosine Kinase. J.Med.Chem., 62, 2019
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8HTR
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![BU of 8htr by Molmil](/molmil-images/mine/8htr) | Crystal structure of Bcl2 in complex with S-9c | Descriptor: | 4-[4-[(2~{S})-2-(2-chlorophenyl)pyrrolidin-1-yl]phenyl]-~{N}-[3-nitro-4-(oxan-4-ylmethylamino)phenyl]sulfonyl-2-(1~{H}-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide, Apoptosis regulator Bcl-2 | Authors: | Liu, J, Xu, M, Feng, Y, Liu, Y. | Deposit date: | 2022-12-21 | Release date: | 2024-05-15 | Last modified: | 2024-06-05 | Method: | X-RAY DIFFRACTION (1.6 Å) | Cite: | Discovery of the Clinical Candidate Sonrotoclax (BGB-11417), a Highly Potent and Selective Inhibitor for Both WT and G101V Mutant Bcl-2. J.Med.Chem., 67, 2024
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8HTS
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![BU of 8hts by Molmil](/molmil-images/mine/8hts) | Crystal structure of Bcl2 in complex with S-10r | Descriptor: | 4-[2-[(2~{S})-2-(2-cyclopropylphenyl)pyrrolidin-1-yl]-7-azaspiro[3.5]nonan-7-yl]-~{N}-[3-nitro-4-(oxan-4-ylmethylamino)phenyl]sulfonyl-2-(1~{H}-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide, Apoptosis regulator Bcl-2 | Authors: | Liu, J, Xu, M, Feng, Y, Liu, Y. | Deposit date: | 2022-12-21 | Release date: | 2024-05-15 | Last modified: | 2024-06-05 | Method: | X-RAY DIFFRACTION (1.25 Å) | Cite: | Discovery of the Clinical Candidate Sonrotoclax (BGB-11417), a Highly Potent and Selective Inhibitor for Both WT and G101V Mutant Bcl-2. J.Med.Chem., 67, 2024
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5H1D
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![BU of 5h1d by Molmil](/molmil-images/mine/5h1d) | Crystal structure of C-terminal of RhoGDI2 | Descriptor: | Rho GDP-dissociation inhibitor 2 | Authors: | Liu, J. | Deposit date: | 2016-10-08 | Release date: | 2016-10-26 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (1.494 Å) | Cite: | NMR characterization of weak interactions between RhoGDI2 and fragment screening hits. Biochim. Biophys. Acta, 1861, 2017
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5GXT
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![BU of 5gxt by Molmil](/molmil-images/mine/5gxt) | Crystal structure of PigG | Descriptor: | MAGNESIUM ION, Maltose-binding periplasmic protein,PigG | Authors: | Zhang, F, Ran, T, Xu, D, Wang, W. | Deposit date: | 2016-09-20 | Release date: | 2017-07-19 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (2.245 Å) | Cite: | Crystal structure of MBP-PigG fusion protein and the essential function of PigG in the prodigiosin biosynthetic pathway in Serratia marcescens FS14. Int. J. Biol. Macromol., 99, 2017
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5GXV
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![BU of 5gxv by Molmil](/molmil-images/mine/5gxv) | Crystal structure of PigG | Descriptor: | MAGNESIUM ION, Maltose-binding periplasmic protein,PigG | Authors: | Zhang, F, Ran, T, Xu, D, Wang, W. | Deposit date: | 2016-09-20 | Release date: | 2017-07-19 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Crystal structure of MBP-PigG fusion protein and the essential function of PigG in the prodigiosin biosynthetic pathway in Serratia marcescens FS14. Int. J. Biol. Macromol., 99, 2017
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4M24
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![BU of 4m24 by Molmil](/molmil-images/mine/4m24) | Crystal structure of the endo-1,4-glucanase, RBcel1, in complex with cellobiose | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Endoglucanase, beta-D-glucopyranose-(1-4)-beta-D-glucopyranose | Authors: | Delsaute, M, Berlemont, R, Van elder, D, Galleni, M, Bauvois, C. | Deposit date: | 2013-08-05 | Release date: | 2014-12-31 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (1.386 Å) | Cite: | Characterisation of two GH family 5 cellulases required for bacterial cellulose production To be Published
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8F7T
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![BU of 8f7t by Molmil](/molmil-images/mine/8f7t) | Glycan-Base ConC Env Trimer | Descriptor: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-6)-2-acetamido-2-deoxy-beta-D-glucopyranose, HIV-1 Env gp120, ... | Authors: | Olia, A.S, Kwong, P.D. | Deposit date: | 2022-11-20 | Release date: | 2023-09-27 | Method: | ELECTRON MICROSCOPY (4.1 Å) | Cite: | Soluble prefusion-closed HIV-envelope trimers with glycan-covered bases. Iscience, 26, 2023
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7XTQ
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![BU of 7xtq by Molmil](/molmil-images/mine/7xtq) | Cryo-EM structure of the R399-bound GPBAR-Gs complex | Descriptor: | G-protein coupled bile acid receptor 1, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1, ... | Authors: | Ma, L, Yang, F, Wu, X, Mao, C, Sun, J, Yu, X, Zhang, Y, Zhang, P. | Deposit date: | 2022-05-17 | Release date: | 2022-07-06 | Last modified: | 2022-08-03 | Method: | ELECTRON MICROSCOPY (3.2 Å) | Cite: | Structural basis and molecular mechanism of biased GPBAR signaling in regulating NSCLC cell growth via YAP activity. Proc.Natl.Acad.Sci.USA, 119, 2022
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