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8I2B

Human SIRT6 in complex with inhibitor 7702

Summary for 8I2B
Entry DOI10.2210/pdb8i2b/pdb
DescriptorNAD-dependent protein deacylase sirtuin-6, TETRAETHYLENE GLYCOL, N1-[[4-(4-aminophenyl)sulfanyl-3-(trifluoromethyl)phenyl]methoxy]benzene-1,4-dicarboxamide, ... (7 entities in total)
Functional Keywordslyase-inhibitor complex, lyase/inhibitor
Biological sourceHomo sapiens (human)
Total number of polymer chains2
Total formula weight67761.58
Authors
Wang, Y. (deposition date: 2023-01-14, release date: 2024-01-17)
Primary citationWang, Y.
The SIRT6 in complex with inhibitor 7702
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.2 Å)
Structure validation

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PDB entries from 2024-05-01

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