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8I0M

Structure of CDK6 in complex with inhibitor

Summary for 8I0M
Entry DOI10.2210/pdb8i0m/pdb
DescriptorCyclin-dependent kinase 6, 2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{N},~{N}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamide (2 entities in total)
Functional Keywordscdk6, inhibitor, complex, cell cycle, cell cycle-inhibitor complex, cell cycle/inhibitor
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight34560.84
Authors
Jiang, C.,Ye, Y.,Huang, Y. (deposition date: 2023-01-11, release date: 2024-01-24)
Primary citationJiang, C.,Ye, Y.,Huang, Y.
Structure of CDK6 in complex with inhibitor
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.7772 Å)
Structure validation

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