Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

7MLC

PYL10 bound to the ABA pan-antagonist 4a

Summary for 7MLC
Entry DOI10.2210/pdb7mlc/pdb
DescriptorAbscisic acid receptor PYL10, GLYCEROL, 1-{2-[3,5-dicyclopropyl-4-(4-{[(quinoxaline-2-carbonyl)amino]methyl}-1H-1,2,3-triazol-1-yl)phenyl]acetamido}cyclohexane-1-carboxylic acid, ... (4 entities in total)
Functional Keywordspyr/pyl/rcar, pyl10, hormone receptor, plant protein, plant protein-antagonist complex, plant protein/antagonist
Biological sourceArabidopsis thaliana (Mouse-ear cress)
Total number of polymer chains1
Total formula weight18433.08
Authors
Peterson, F.C.,Vaidya, A.S.,Volkman, B.F.,Cutler, S.R. (deposition date: 2021-04-28, release date: 2021-09-29, Last modification date: 2023-10-18)
Primary citationVaidya, A.S.,Peterson, F.C.,Eckhardt, J.,Xing, Z.,Park, S.Y.,Dejonghe, W.,Takeuchi, J.,Pri-Tal, O.,Faria, J.,Elzinga, D.,Volkman, B.F.,Todoroki, Y.,Mosquna, A.,Okamoto, M.,Cutler, S.R.
Click-to-lead design of a picomolar ABA receptor antagonist with potent activity in vivo.
Proc.Natl.Acad.Sci.USA, 118:-, 2021
Cited by
PubMed: 34531324
DOI: 10.1073/pnas.2108281118
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.77 Å)
Structure validation

218853

PDB entries from 2024-04-24

PDB statisticsPDBj update infoContact PDBjnumon