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6Q55

Crystal structure of Cryptosporidium hominis CPSF3 in complex with Compound 61

Summary for 6Q55
Entry DOI10.2210/pdb6q55/pdb
DescriptorCleavage and Polyadenylation Specificity Factor 3 (CPSF3), ZINC ION, 3-[7,7-bis(oxidanyl)-8-oxa-7-boranuidabicyclo[4.3.0]nona-1(6),2,4-trien-5-yl]propanoic acid, ... (7 entities in total)
Functional Keywordsmrna processing factor, metallo-beta-lactamase, beta-casp, oxaborole-inhibitor, rna binding protein
Biological sourceCryptosporidium hominis TU502
Total number of polymer chains1
Total formula weight55113.32
Authors
Palencia, A.,Swale, C. (deposition date: 2018-12-07, release date: 2019-11-20, Last modification date: 2024-01-24)
Primary citationSwale, C.,Bougdour, A.,Gnahoui-David, A.,Tottey, J.,Georgeault, S.,Laurent, F.,Palencia, A.,Hakimi, M.A.
Metal-captured inhibition of pre-mRNA processing activity by CPSF3 controls Cryptosporidium infection.
Sci Transl Med, 11:-, 2019
Cited by
PubMed: 31694928
DOI: 10.1126/scitranslmed.aax7161
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2 Å)
Structure validation

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