6M9H
JAK2 JH2 in complex with diaminopyrimidine JAK040
Summary for 6M9H
Entry DOI | 10.2210/pdb6m9h/pdb |
Descriptor | Tyrosine-protein kinase JAK2, 4-({4-amino-6-[4-(2-hydroxyethyl)-1H-imidazol-1-yl]pyrimidin-2-yl}amino)benzonitrile, GLYCEROL, ... (5 entities in total) |
Functional Keywords | transferase/transferase inhibitor, transferase, transferase-transferase inhibitor complex |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 33612.53 |
Authors | Puleo, D.E.,Schlessinger, J.,Jorgensen, W.L. (deposition date: 2018-08-23, release date: 2018-09-05, Last modification date: 2024-03-13) |
Primary citation | Puleo, D.E.,Schlessinger, J. JAK2 JH2 Binders To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.79 Å) |
Structure validation
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