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6L04

Crystal structure of uPA_H99Y in complex with 31F

Summary for 6L04
Entry DOI10.2210/pdb6l04/pdb
DescriptorUrokinase-type plasminogen activator, 3-azanyl-5-(azepan-1-yl)-N-carbamimidoyl-6-(2,4-dimethoxypyrimidin-5-yl)pyrazine-2-carboxamide (3 entities in total)
Functional Keywordsurokinase, amiloride, hydrolase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight28026.90
Authors
Buckley, B.,Jiang, L.G.,Huang, M.D.,Kelso, M.,Ranson, M. (deposition date: 2019-09-26, release date: 2020-09-30, Last modification date: 2023-11-22)
Primary citationBuckley, B.,Jiang, L.G.,Huang, M.D.,Kelso, M.,Ranson, M.
Crystal structure of uPA_H99Y in complex with 31F
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.21 Å)
Structure validation

221051

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