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6HXR

Human PARP16 (ARTD15) IN COMPLEX WITH EB-47

Summary for 6HXR
Entry DOI10.2210/pdb6hxr/pdb
DescriptorMono [ADP-ribose] polymerase PARP16, 2-[4-[(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]carbonylpiperazin-1-yl]-N-(1-oxidanylidene-2,3-dihydroisoindol-4-yl)ethanamide (2 entities in total)
Functional Keywordstransferase, adp-ribose, parp16, artd15, adp-ribosylation, eb-47, inhibitor complex
Biological sourceHomo sapiens (Human)
Total number of polymer chains3
Total formula weight101821.78
Authors
Karlberg, T.,Pinto, A.F.,Thorsell, A.G.,Schuler, H. (deposition date: 2018-10-18, release date: 2019-10-30, Last modification date: 2024-01-31)
Primary citationKarlberg, T.,Pinto, A.F.,Thorsell, A.G.,Schuler, H.
Human PARP16 (ARTD15) IN COMPLEX WITH EB-47
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.9 Å)
Structure validation

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