6BU6
Crystal Structure of the Human vaccinia-related kinase bound to a bis-difluorophenol-aminopyridine inhibitor
Summary for 6BU6
Entry DOI | 10.2210/pdb6bu6/pdb |
Descriptor | Serine/threonine-protein kinase VRK1, 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol), GLYCEROL, ... (6 entities in total) |
Functional Keywords | transferase, protein kinase domain, structural genomics, structural genomics consortium, sgc, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 4 |
Total formula weight | 166388.43 |
Authors | Counago, R.M.,dos Reis, C.V.,de Souza, G.P.,Santiago, A.S.,Azevedo, A.,Guimaraes, C.,Mascarello, A.,Gama, F.,Ferreira, M.,Massirer, K.B.,Arruda, P.,Edwards, A.M.,Elkins, J.M.,Structural Genomics Consortium (SGC) (deposition date: 2017-12-08, release date: 2017-12-20, Last modification date: 2023-10-04) |
Primary citation | Counago, R.M.,dos Reis, C.V.,de Souza, G.P.,Santiago, A.S.,Azevedo, H.,Guimaraes, C.,Mascarello, A.,Gama, F.,Ferreira, M.,Massirer, K.B.,Arruda, P.,Edwards, A.M.,Elkins, J.M.,Structural Genomics Consortium (SGC) Crystal Structure of the Human vaccinia-related kinase bound to a bis-difluorophenol-aminopyridine inhibitor To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.8 Å) |
Structure validation
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