5H1T
Complex structure of TRIM24 PHD-bromodomain and inhibitor 1
Summary for 5H1T
Entry DOI | 10.2210/pdb5h1t/pdb |
Related | 5H1U 5H1V |
Descriptor | Transcription intermediary factor 1-alpha, ZINC ION, methyl 6-azanyl-3,4-dihydro-2H-quinoline-1-carboxylate, ... (5 entities in total) |
Functional Keywords | transcription, transcription inhibitor, transcription-transcription inhibitor complex, transcription/transcription inhibitor |
Biological source | Homo sapiens (Human) |
Cellular location | Nucleus : O15164 |
Total number of polymer chains | 4 |
Total formula weight | 86429.77 |
Authors | |
Primary citation | Liu, J.,Li, F.,Bao, H.,Jiang, Y.,Zhang, S.,Ma, R.,Gao, J.,Wu, J.,Ruan, K. The polar warhead of a TRIM24 bromodomain inhibitor rearranges a water-mediated interaction network FEBS J., 284:1082-1095, 2017 Cited by PubMed: 28207202DOI: 10.1111/febs.14041 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.951 Å) |
Structure validation
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