5H1E
Interaction between vitamin D receptor and coactivator peptide SRC2-3
Summary for 5H1E
Entry DOI | 10.2210/pdb5h1e/pdb |
Descriptor | Vitamin D3 receptor, Nuclear receptor coactivator 2 peptide, 5-{2-[1-(5-HYDROXY-1,5-DIMETHYL-HEXYL)-7A-METHYL-OCTAHYDRO-INDEN-4-YLIDENE]-ETHYLIDENE}-4-METHYLENE-CYCLOHEXANE-1,3-DIOL, ... (4 entities in total) |
Functional Keywords | transcription, vitamin d3, vdre, rxr, co-factors, tif2 |
Biological source | Rattus norvegicus (Rat) More |
Total number of polymer chains | 2 |
Total formula weight | 32605.52 |
Authors | Egawa, D.,Itoh, T.,Kato, A.,Kataoka, S.,Anami, Y.,Yamamoto, K. (deposition date: 2016-10-08, release date: 2017-01-11, Last modification date: 2024-03-20) |
Primary citation | Egawa, D.,Itoh, T.,Kato, A.,Kataoka, S.,Anami, Y.,Yamamoto, K. SRC2-3 binds to vitamin D receptor with high sensitivity and strong affinity Bioorg. Med. Chem., 25:568-574, 2017 Cited by PubMed: 27890450DOI: 10.1016/j.bmc.2016.11.020 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.6 Å) |
Structure validation
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