5C67
Human Mesotrypsin in complex with amyloid precursor protein inhibitor variant APPI-M17G/I18F/F34V
Summary for 5C67
Entry DOI | 10.2210/pdb5c67/pdb |
Descriptor | Trypsin-3, Amyloid beta A4 protein (3 entities in total) |
Functional Keywords | appi, kunitz domain, trypsin, hyrdolase-hydrolase inhibitor complex, hyrdolase/hydrolase inhibitor |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 4 |
Total formula weight | 66784.71 |
Authors | Kayode, O.,Sankaran, B.,Radisky, E.S. (deposition date: 2015-06-22, release date: 2016-05-04, Last modification date: 2023-09-27) |
Primary citation | Cohen, I.,Kayode, O.,Hockla, A.,Sankaran, B.,Radisky, D.C.,Radisky, E.S.,Papo, N. Combinatorial protein engineering of proteolytically resistant mesotrypsin inhibitors as candidates for cancer therapy. Biochem.J., 473:1329-1341, 2016 Cited by PubMed: 26957636DOI: 10.1042/BJ20151410 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.83 Å) |
Structure validation
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