4XSX
Crystal structure of CBR 703 bound to Escherichia coli RNA polymerase holoenzyme
Summary for 4XSX
Entry DOI | 10.2210/pdb4xsx/pdb |
Related | 4XSY 4XSZ |
Descriptor | DNA-directed RNA polymerase subunit alpha, DNA-directed RNA polymerase subunit beta, DNA-directed RNA polymerase subunit beta', ... (8 entities in total) |
Functional Keywords | bacterial rna polymerase antibiotic complex, transcription-antibiotic complex, transcription/antibiotic |
Biological source | Escherichia coli (strain K12) More |
Cellular location | Cytoplasm : P00579 |
Total number of polymer chains | 12 |
Total formula weight | 860212.15 |
Authors | Bae, B.,Darst, S.A. (deposition date: 2015-01-22, release date: 2015-07-22, Last modification date: 2023-09-27) |
Primary citation | Bae, B.,Nayak, D.,Ray, A.,Mustaev, A.,Landick, R.,Darst, S.A. CBR antimicrobials inhibit RNA polymerase via at least two bridge-helix cap-mediated effects on nucleotide addition. Proc.Natl.Acad.Sci.USA, 112:E4178-E4187, 2015 Cited by PubMed: 26195788DOI: 10.1073/pnas.1502368112 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.708 Å) |
Structure validation
Download full validation report