4WM9
Acinetobacter baumanii OXA-24 complex with Avibactam
Summary for 4WM9
Entry DOI | 10.2210/pdb4wm9/pdb |
Related | 2JC7 |
Descriptor | Beta-lactamase, (2S,5R)-1-formyl-5-[(sulfooxy)amino]piperidine-2-carboxamide, SULFATE ION, ... (6 entities in total) |
Functional Keywords | beta-lactamase, class d carbapenemase, inhibitor, hydrolase |
Biological source | Acinetobacter baumannii |
Total number of polymer chains | 1 |
Total formula weight | 28408.50 |
Authors | Mangani, S.,Benvenuti, M.,Docquier, J.-D. (deposition date: 2014-10-08, release date: 2014-12-03, Last modification date: 2024-01-10) |
Primary citation | Lahiri, S.D.,Mangani, S.,Jahic, H.,Benvenuti, M.,Durand-Reville, T.F.,De Luca, F.,Ehmann, D.E.,Rossolini, G.M.,Alm, R.A.,Docquier, J.D. Molecular Basis of Selective Inhibition and Slow Reversibility of Avibactam against Class D Carbapenemases: A Structure-Guided Study of OXA-24 and OXA-48. Acs Chem.Biol., 10:591-600, 2015 Cited by PubMed: 25406838DOI: 10.1021/cb500703p PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.4 Å) |
Structure validation
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