4U7G
Oxidized quinone reductase 2 in complex with CK2 inhibitor TBBz
Summary for 4U7G
Entry DOI | 10.2210/pdb4u7g/pdb |
Related | 4U7F 4U7H |
Descriptor | Ribosyldihydronicotinamide dehydrogenase [quinone], ZINC ION, FLAVIN-ADENINE DINUCLEOTIDE, ... (5 entities in total) |
Functional Keywords | quinone reductase 2, ck2 inhibitor, oxidoreductase-inhibitor complex, oxidoreductase/inhibitor |
Biological source | Homo sapiens (Human) |
Cellular location | Cytoplasm: P16083 |
Total number of polymer chains | 2 |
Total formula weight | 54268.03 |
Authors | Leung, K.K.,Shilton, B.H. (deposition date: 2014-07-30, release date: 2015-02-11, Last modification date: 2023-09-27) |
Primary citation | Leung, K.K.,Shilton, B.H. Quinone Reductase 2 Is an Adventitious Target of Protein Kinase CK2 Inhibitors TBBz (TBI) and DMAT. Biochemistry, 54:47-59, 2015 Cited by PubMed: 25379648DOI: 10.1021/bi500959t PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.96 Å) |
Structure validation
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