4QQE
Crystal structure of WDR5, WD repeat domain 5 in complex with compound SGC-DS-MT-0345
Summary for 4QQE
Entry DOI | 10.2210/pdb4qqe/pdb |
Descriptor | WD repeat-containing protein 5, N-[2-(4-methylpiperazin-1-yl)-5-(quinolin-3-yl)phenyl]-6-oxo-4-(trifluoromethyl)-1,6-dihydropyridine-3-carboxamide, CHLORIDE ION, ... (6 entities in total) |
Functional Keywords | wdr5, structural genomics, structural genomics consortium, sgc, transcription |
Biological source | Homo sapiens (human) |
Cellular location | Nucleus : P61964 |
Total number of polymer chains | 1 |
Total formula weight | 35019.05 |
Authors | Dong, A.,Dombrovski, L.,Wernimont, A.,Smil, D.,Getlik, M.,Senisterra, G.,Poda, G.,Al-Awar, R.,Bountra, C.,Arrowsmith, C.H.,Edwards, A.M.,Brown, P.J.,Schapira, M.,Vedadi, M.,Wu, H.,Structural Genomics Consortium (SGC) (deposition date: 2014-06-27, release date: 2014-07-30, Last modification date: 2023-09-20) |
Primary citation | Dombrovski, L.,Dong, A.,Wernimont, A.,Smil, D.,Getlik, M.,Senisterra, G.,Poda, G.,Al-Awar, R.,Bountra, C.,Arrowsmith, C.H.,Edwards, A.M.,Brown, P.J.,Schapira, M.,Vedadi, M.,Wu, H. Crystal structure of WDR5, WD repeat domain 5 in complex with compound SGC-DS-MT-0345 To be Published, |
Experimental method | X-RAY DIFFRACTION (1.8 Å) |
Structure validation
Download full validation report