4MY6
EnaH-EVH1 in complex with peptidomimetic low-molecular weight inhibitor Ac-[2-Cl-F]-[ProM-2]-[ProM-1]-OH
Summary for 4MY6
Entry DOI | 10.2210/pdb4my6/pdb |
Related PRD ID | PRD_001198 |
Descriptor | Protein enabled homolog, (3aR,5aS,8S,10aS)-1-[(3S,6R,8aS)-1'-[(2S)-2-acetamido-3-(2-chlorophenyl)propanoyl]-5-oxidanylidene-spiro[1,2,3,8a-tetrahydroindolizine-6,2'-pyrrolidine]-3-yl]carbonyl-10-oxidanylidene-2,3,3a,5a,8,10a-hexahydrodipyrrolo[3,2-b:3',1'-f]azepine-8-carboxylic acid, BROMIDE ION, ... (4 entities in total) |
Functional Keywords | molecular recognition, actin dynamics, cell adhesion-inhibitor complex, cell adhesion/inhibitor |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm: Q8N8S7 |
Total number of polymer chains | 2 |
Total formula weight | 26768.67 |
Authors | Barone, M.,Roske, Y.,Kuehne, R. (deposition date: 2013-09-27, release date: 2014-10-15, Last modification date: 2023-09-20) |
Primary citation | Opitz, R.,Muller, M.,Reuter, C.,Barone, M.,Soicke, A.,Roske, Y.,Piotukh, K.,Huy, P.,Beerbaum, M.,Wiesner, B.,Beyermann, M.,Schmieder, P.,Freund, C.,Volkmer, R.,Oschkinat, H.,Schmalz, H.G.,Kuhne, R. A modular toolkit to inhibit proline-rich motif-mediated protein-protein interactions. Proc.Natl.Acad.Sci.USA, 112:5011-5016, 2015 Cited by PubMed: 25848013DOI: 10.1073/pnas.1422054112 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.7 Å) |
Structure validation
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