3WPN
Kinesin spindle protein Eg5 in complex with ATP-competitive inhibitor PVZB1194
Summary for 3WPN
Entry DOI | 10.2210/pdb3wpn/pdb |
Related | 1II6 1Q0B 3ZCW |
Descriptor | Kinesin-like protein KIF11, 3'-fluoro-4'-(trifluoromethyl)biphenyl-4-sulfonamide (3 entities in total) |
Functional Keywords | cell cycle, motor domain, atp binding |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm : P52732 |
Total number of polymer chains | 1 |
Total formula weight | 43194.91 |
Authors | Yokoyama, H.,Katoh, S.,Fujii, S. (deposition date: 2014-01-14, release date: 2015-01-21, Last modification date: 2023-11-08) |
Primary citation | Yokoyama, H.,Sawada, J.,Katoh, S.,Matsuno, K.,Ogo, N.,Ishikawa, Y.,Hashimoto, H.,Fujii, S.,Asai, A. Structural basis of new allosteric inhibition in Kinesin spindle protein eg5 Acs Chem.Biol., 10:1128-1136, 2015 Cited by PubMed: 25622007DOI: 10.1021/cb500939x PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.8 Å) |
Structure validation
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