3WMH
Human PPAR gamma ligand binding domain in complex with a gammma selective synthetic partial agonist MEKT75
Summary for 3WMH
Entry DOI | 10.2210/pdb3wmh/pdb |
Related | 3vso 3vsp |
Descriptor | Peroxisome proliferator-activated receptor gamma, N-(phenylsulfonyl)-4-propoxy-3-({[4-(pyrimidin-2-yl)benzoyl]amino}methyl)benzamide (3 entities in total) |
Functional Keywords | mainly alpha, nuclear receptor, transcription |
Biological source | Homo sapiens (human) |
Cellular location | Nucleus: P37231 |
Total number of polymer chains | 2 |
Total formula weight | 66122.49 |
Authors | Oyama, T.,Ohashi, M.,Miyachi, H.,Kusunoki, M. (deposition date: 2013-11-19, release date: 2014-11-19, Last modification date: 2023-11-08) |
Primary citation | Oyama, T.,Ohashi, M.,Miyachi, H.,Kusunoki, M. Human PPRR gamma ligand binding domain in complex with a gammma selective synthetic partial agonist MEKT75 TO BE PUBLISHED, |
Experimental method | X-RAY DIFFRACTION (2.1 Å) |
Structure validation
Download full validation report