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3VSP

Human PPAR gamma ligand binding domain in complex with a gamma selective agonist mekt28

Summary for 3VSP
Entry DOI10.2210/pdb3vsp/pdb
Related3VSO 3an3
DescriptorPeroxisome proliferator-activated receptor gamma, (2R)-2-benzyl-3-[3-({[4-(piperidin-1-yl)benzoyl]amino}methyl)-4-propoxyphenyl]propanoic acid (3 entities in total)
Functional Keywordsmainly alpha, nuclear receptor, transcription
Biological sourceHomo sapiens (human)
Cellular locationNucleus: P37231
Total number of polymer chains2
Total formula weight65575.96
Authors
Oyama, T.,Waku, T.,Ohashi, M.,Morikawa, K.,Miyachi, H. (deposition date: 2012-04-30, release date: 2013-05-01, Last modification date: 2023-11-08)
Primary citationOyama, T.,Waku, T.,Ohashi, M.,Morikawa, K.,Miyachi, H.
Human PPAR gamma ligand binding domain in complex with a gamma selective agonist mekt28
To be Published,
Experimental method
X-RAY DIFFRACTION (2.4 Å)
Structure validation

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