3RAW
Crystal Structure of human CDC-like kinase 3 isoform in complex with leucettine L41
Summary for 3RAW
Entry DOI | 10.2210/pdb3raw/pdb |
Related | 2EU9 |
Descriptor | Dual specificity protein kinase CLK3, 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4H-imidazol-4-one (3 entities in total) |
Functional Keywords | transferase, kinase, tyrosine-protein kinase, serine/threonine-protein kinase, nucleotide-binding, structural genomics consortium, sgc |
Biological source | Homo sapiens (human) |
Cellular location | Nucleus: P49761 |
Total number of polymer chains | 2 |
Total formula weight | 90194.73 |
Authors | Filippakopoulos, P.,Fedorov, O.,King, O.,Debdab, M.,Carreaux, F.,Renault, S.,Bullock, A.,Muniz, J.R.C.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Weigelt, J.,Bountra, C.,Meijer, L.,Bazureau, J.P.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2011-03-28, release date: 2011-05-04, Last modification date: 2023-09-13) |
Primary citation | Filippakopoulos, P.,Fedorov, O.,King, O.,Bullock, A.,Muniz, J.R.C.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Weigelt, J.,Bountra, C.,Knapp, S.,Structural Genomics Consortium (SGC) Crystal Structure of human CDC-like kinase 3 isoform with a benzo-dioxol ligand To be Published, |
Experimental method | X-RAY DIFFRACTION (2.09 Å) |
Structure validation
Download full validation report