3FY0
Crystal structure of PAK1 kinase domain with ruthenium complex DW1
Summary for 3FY0
Entry DOI | 10.2210/pdb3fy0/pdb |
Related | 3FXZ |
Descriptor | Serine/threonine-protein kinase PAK 1, Ruthenium pyridocarbazole (3 entities in total) |
Functional Keywords | transferase, kinase, atp-binding, phosphorylation, allosteric enzyme, apoptosis, cell junction, nucleotide-binding, phosphoprotein, serine/threonine-protein kinase |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm : Q13153 |
Total number of polymer chains | 1 |
Total formula weight | 33863.68 |
Authors | Maksimoska, J.,Marmorstein, R.,Meggers, E. (deposition date: 2009-01-21, release date: 2009-03-03, Last modification date: 2021-10-20) |
Primary citation | Maksimoska, J.,Feng, L.,Harms, K.,Yi, C.,Kissil, J.,Marmorstein, R.,Meggers, E. Targeting Large Kinase Active Site with Rigid, Bulky Octahedral Ruthenium Complexes J.Am.Chem.Soc., 130:15764-15765, 2008 Cited by PubMed: 18973295PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.35 Å) |
Structure validation
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