2J0F
Structural basis for non-competitive product inhibition in human thymidine phosphorylase: implication for drug design
Summary for 2J0F
Entry DOI | 10.2210/pdb2j0f/pdb |
Related | 1UOU |
Descriptor | THYMIDINE PHOSPHORYLASE, THYMINE (3 entities in total) |
Functional Keywords | htp, chemotaxis, transferase, polymorphism, disease mutation, glycosyltransferase, angiogenesis, growth factor, differentiation, developmental protein, human thymidine phosphorylase |
Biological source | HOMO SAPIENS (HUMAN) |
Total number of polymer chains | 4 |
Total formula weight | 200499.86 |
Authors | El Omari, K.,Bronckaers, A.,Liekens, S.,Perez-Perez, M.J.,Balzarini, J.,Stammers, D.K. (deposition date: 2006-08-02, release date: 2006-10-11, Last modification date: 2023-12-13) |
Primary citation | El Omari, K.,Bronckaers, A.,Liekens, S.,Perez-Perez, M.,Balzarini, J.,Stammers, D.K. Structural Basis for Non-Competitive Product Inhibition in Human Thymidine Phosphorylase: Implications for Drug Design. Biochem.J., 399:199-, 2006 Cited by PubMed: 16803458DOI: 10.1042/BJ20060513 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.31 Å) |
Structure validation
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