2IZU
Structure of casein kinase gamma 3 in complex with inhibitor
Summary for 2IZU
Entry DOI | 10.2210/pdb2izu/pdb |
Related | 2CHL 2IUR 2IZS 2IZT |
Descriptor | CASEIN KINASE I ISOFORM GAMMA-3, 2-({6-[(3-CHLOROPHENYL)AMINO]-9-ISOPROPYL-9H-PURIN-2-YL}AMINO)-3-METHYLBUTAN-1-OL, 1,2-ETHANEDIOL, ... (5 entities in total) |
Functional Keywords | serine/threonine-protein kinase, kinase, transferase, atp- binding, phosphorylation, nucleotide-binding, wnt signaling pathway, serine/threonine kinase |
Biological source | HOMO SAPIENS (HUMAN) |
Cellular location | Cytoplasm: Q9Y6M4 |
Total number of polymer chains | 1 |
Total formula weight | 39103.33 |
Authors | Bunkoczi, G.,Salah, E.,Rellos, P.,Das, S.,Fedorov, O.,Savitsky, P.,Debreczeni, J.E.,Gileadi, O.,Sundstrom, M.,Edwards, A.,Arrowsmith, C.,Weigelt, J.,von Delft, F.,Knapp, S. (deposition date: 2006-07-26, release date: 2006-08-01, Last modification date: 2023-12-13) |
Primary citation | Bunkoczi, G.,Salah, E.,Rellos, P.,Das, S.,Fedorov, O.,Savitsky, P.,Debreczeni, J.E.,Gileadi, O.,Sundstrom, M.,Edwards, A.,Arrowsmith, C.,Weigelt, J.,von Delft, F.,Knapp, S. Inhibitor Binding by Casein Kinases To be Published, |
Experimental method | X-RAY DIFFRACTION (1.85 Å) |
Structure validation
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