2EXC
Inhibitor complex of JNK3
Summary for 2EXC
Entry DOI | 10.2210/pdb2exc/pdb |
Descriptor | Mitogen-activated protein kinase 10, N-{2'-[(4-FLUOROPHENYL)AMINO]-4,4'-BIPYRIDIN-2-YL}-4-METHOXYCYCLOHEXANECARBOXAMIDE (3 entities in total) |
Functional Keywords | enzyme-inhibitor complex, kinase inhibitor, transferase |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm: P53779 |
Total number of polymer chains | 1 |
Total formula weight | 41601.12 |
Authors | |
Primary citation | Swahn, B.-M.,Xue, Y.,Arzel, E.,Kallin, E.,Magnus, A.,Plobeck, N.,Viklund, J. Inhibitor complex of JNK3 To be Published, |
Experimental method | X-RAY DIFFRACTION (2.75 Å) |
Structure validation
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