1YAT
IMPROVED CALCINEURIN INHIBITION BY YEAST FKBP12-DRUG COMPLEXES. CRYSTALLOGRAPHIC AND FUNCTIONAL ANALYSIS
Summary for 1YAT
Entry DOI | 10.2210/pdb1yat/pdb |
Descriptor | FK506 BINDING PROTEIN, 8-DEETHYL-8-[BUT-3-ENYL]-ASCOMYCIN (3 entities in total) |
Functional Keywords | binding protein |
Biological source | Saccharomyces cerevisiae (baker's yeast) |
Cellular location | Cytoplasm: P20081 |
Total number of polymer chains | 1 |
Total formula weight | 12842.65 |
Authors | Rotonda, J.,Becker, J.W. (deposition date: 1993-01-06, release date: 1993-10-31, Last modification date: 2024-02-14) |
Primary citation | Rotonda, J.,Burbaum, J.J.,Chan, H.K.,Marcy, A.I.,Becker, J.W. Improved calcineurin inhibition by yeast FKBP12-drug complexes. Crystallographic and functional analysis. J.Biol.Chem., 268:7607-7609, 1993 Cited by PubMed: 7681823PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.5 Å) |
Structure validation
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