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1VJB

crystal structure of the ligand-binding domain of the estrogen-related receptor gamma in complex with 4-hydroxytamoxifen

Summary for 1VJB
Entry DOI10.2210/pdb1vjb/pdb
Related1KV6
DescriptorEstrogen-related receptor gamma, 4-HYDROXYTAMOXIFEN (2 entities in total)
Functional Keywordsligand-binding domain, antagonist complex, transcription
Biological sourceMus musculus (Mouse)
Total number of polymer chains2
Total formula weight57548.91
Authors
Greschik, H.,Flaig, R.,Renaud, J.P.,Moras, D. (deposition date: 2004-02-03, release date: 2004-06-08, Last modification date: 2023-08-23)
Primary citationGreschik, H.,Flaig, R.,Renaud, J.P.,Moras, D.
Structural Basis for the Deactivation of the Estrogen-related Receptor {gamma} by Diethylstilbestrol or 4-Hydroxytamoxifen and Determinants of Selectivity.
J.Biol.Chem., 279:33639-33646, 2004
Cited by
PubMed: 15161930
DOI: 10.1074/jbc.M402195200
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (3.2 Å)
Structure validation

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