1PYX
GSK-3 Beta complexed with AMP-PNP
Summary for 1PYX
Entry DOI | 10.2210/pdb1pyx/pdb |
Descriptor | Glycogen synthase kinase-3 beta, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ... (4 entities in total) |
Functional Keywords | kinase, insulin pathway, transferase |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm: P49841 |
Total number of polymer chains | 2 |
Total formula weight | 95020.38 |
Authors | Bertrand, J.A.,Thieffine, S.,Vulpetti, A.,Cristiani, C.,Valsasina, B.,Knapp, S.,Kalisz, H.M.,Flocco, M. (deposition date: 2003-07-09, release date: 2003-10-21, Last modification date: 2023-08-16) |
Primary citation | Bertrand, J.A.,Thieffine, S.,Vulpetti, A.,Cristiani, C.,Valsasina, B.,Knapp, S.,Kalisz, H.M.,Flocco, M. Structural characterization of the GSK-3beta active site using selective and non-selective ATP-mimetic inhibitors J.Mol.Biol., 333:393-407, 2003 Cited by PubMed: 14529625DOI: 10.1016/j.jmb.2003.08.031 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.4 Å) |
Structure validation
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