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7WVU

Cryo-EM structure of the human formyl peptide receptor 1 in complex with fMLF and Gi1

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1RfMet-Leu-Phe receptorpolymer37140754.71UniProt (P21462)
Pfam (PF00001)
In PDB
Homo sapiens (human)fMLP receptor,N-formyl peptide receptor,FPR,N-formylpeptide chemoattractant receptor
2AGuanine nucleotide-binding protein G(i) subunit alpha-1polymer35440447.11UniProt (P63096)
Pfam (PF00503)
In PDB
Homo sapiens (human)Adenylate cyclase-inhibiting G alpha protein
3BGuanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1polymer35138744.41UniProt (P62873)
Pfam (PF00400)
In PDB
Homo sapiens (human)Transducin beta chain 1
4CGuanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2polymer717861.11UniProt (P59768)
Pfam (PF00631)
In PDB
Homo sapiens (human)G gamma-I
5LFME-LEU-PHEpolymer3437.61Homo sapiens
Sequence modifications
R: 2 - 321 (UniProt: P21462)
PDBExternal DatabaseDetails
Gly -1-expression tag
Ala 0-expression tag
Pro 1-expression tag
Glu 322-expression tag
Phe 323-expression tag
Leu 324-expression tag
Glu 325-expression tag
Val 326-expression tag
Leu 327-expression tag
Phe 328-expression tag
Gln 329-expression tag
Gly 330-expression tag
Pro 331-expression tag
Gly 332-expression tag
Ser 333-expression tag
Trp 334-expression tag
Ser 335-expression tag
His 336-expression tag
Pro 337-expression tag
Gln 338-expression tag
Phe 339-expression tag
Glu 340-expression tag
Lys 341-expression tag
Gly 342-expression tag
Ser 343-expression tag
Gly 344-expression tag
Ala 345-expression tag
Gly 346-expression tag
Ala 347-expression tag
Ser 348-expression tag
Ala 349-expression tag
Gly 350-expression tag
Ser 351-expression tag
Trp 352-expression tag
Ser 353-expression tag
His 354-expression tag
Pro 355-expression tag
Gln 356-expression tag
Phe 357-expression tag
Glu 358-expression tag
Lys 359-expression tag
Gly 360-expression tag
Ser 361-expression tag
Asp 362-expression tag
Tyr 363-expression tag
Lys 364-expression tag
Asp 365-expression tag
Asp 366-expression tag
Asp 367-expression tag
Asp 368-expression tag
Lys 369-expression tag
A: 1 - 354 (UniProt: P63096)
PDBExternal DatabaseDetails
Cys 47Ser 47engineered mutation
Thr 202Gly 202engineered mutation
Ala 203Gly 203engineered mutation
Ala 245Glu 245engineered mutation
Ser 326Ala 326engineered mutation
B: 2 - 340 (UniProt: P62873)
PDBExternal DatabaseDetails
Met -10-expression tag
His -9-expression tag
His -8-expression tag
His -7-expression tag
His -6-expression tag
His -5-expression tag
His -4-expression tag
Gly -3-expression tag
Ser -2-expression tag
Leu -1-expression tag
Leu 0-expression tag
Gln 1-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains5
Total formula weight128244.9
All*Total formula weight128244.9
*Water molecules are not included.

221051

PDB entries from 2024-06-12

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