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6KJV

Structure of thermal-stabilised(M9) human GLP-1 receptor transmembrane domain

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, BGlucagon-like peptide 1 receptor,Endolysin,Glucagon-like peptide 1 receptorpolymer45552583.32UniProt (P43220)
UniProt (P00720)
Pfam (PF00002)
Pfam (PF00959)
In PDB
Homo sapiens (Human)GLP-1R,Lysis protein,Lysozyme,Muramidase,GLP-1R
2A, BN-{4-[(R)-(3,3-dimethylcyclobutyl)({6-[4-(trifluoromethyl)-1H-imidazol-1-yl]pyridin-3-yl}amino)methyl]benzene-1-carbonyl}-beta-alaninenon-polymer515.52Chemie (97Y)
3A, B(2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoatenon-polymer356.52Chemie (OLC)
4waterwater18.08Chemie (HOH)
Sequence modifications
A, B: 128 - 257 (UniProt: P43220)
PDBExternal DatabaseDetails
Ser 127-expression tag
Cys 193Ser 193engineered mutation
Phe 196Ile 196engineered mutation
-Tyr 205deletion
-Ser 206deletion
-Thr 207deletion
-Ala 208deletion
-Ala 209deletion
-Gln 210deletion
-Gln 211deletion
-His 212deletion
-Gln 213deletion
-Trp 214deletion
Gly 212-linker
Ser 213-linker
Gly 214-linker
Ala 225Ser 225engineered mutation
A, B: 1001 - 1160 (UniProt: P00720)
PDBExternal DatabaseDetails
Gly 1011Arg 12engineered mutation
Thr 1053Cys 54engineered mutation
Ala 1096Cys 97engineered mutation
Arg 1136Ile 137engineered mutation
A, B: 261 - 431 (UniProt: P43220)
PDBExternal DatabaseDetails
Ala 271Ser 271engineered mutation
Cys 317Ile 317engineered mutation
Ile 318Gly 318engineered mutation
Ala 346Lys 346engineered mutation
Phe 347Cys 347engineered mutation
Cys 361Gly 361engineered mutation
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains2
Total formula weight105166.6
Non-Polymers*Number of molecules4
Total formula weight1744.1
All*Total formula weight106910.7
*Water molecules are not included.

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PDB entries from 2024-06-12

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