6BXH
Menin in complex with MI-853
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Menin | polymer | 509 | 56626.5 | 1 | UniProt (O00255) Pfam (PF05053) In PDB | Homo sapiens (Human) | |
2 | A | DIMETHYL SULFOXIDE | non-polymer | 78.1 | 1 | Chemie (DMS) | |||
3 | A | SULFATE ION | non-polymer | 96.1 | 1 | Chemie (SO4) | |||
4 | A | 1-{2-[4-(fluoroacetyl)piperazin-1-yl]ethyl}-4-methyl-5-[(4-{[6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-yl]amino}piperidin-1-yl)methyl]-1H-indole-2-carbonitrile | non-polymer | 656.7 | 1 | Chemie (EE7) | |||
5 | water | water | 18.0 | 129 | Chemie (HOH) |
Sequence modifications
A: 1 - 459 (UniProt: O00255)
PDB | External Database | Details |
---|---|---|
Gly -4 | - | expression tag |
Gly -3 | - | expression tag |
Ser -2 | - | expression tag |
Ser -1 | - | expression tag |
Ser 0 | - | expression tag |
- | Glu 387 | deletion |
- | Glu 388 | deletion |
- | Arg 389 | deletion |
- | Pro 390 | deletion |
- | Gly 391 | deletion |
- | Glu 392 | deletion |
- | Gln 393 | deletion |
- | Ser 394 | deletion |
- | Gln 395 | deletion |
- | Gly 396 | deletion |
- | Thr 397 | deletion |
- | Gln 398 | deletion |
Val 460 | - | expression tag |
Pro 461 | - | expression tag |
Ala 539 | - | expression tag |
Pro 540 | - | expression tag |
Ala 541 | - | expression tag |
Ala 542 | - | expression tag |
Ser 543 | - | expression tag |
Pro 544 | - | expression tag |
Pro 545 | - | expression tag |
Pro 546 | - | expression tag |
Glu 547 | - | expression tag |
Gly 548 | - | expression tag |
Pro 549 | - | expression tag |
Val 550 | - | expression tag |
Leu 551 | - | expression tag |
Thr 552 | - | expression tag |
Phe 553 | - | expression tag |
Gln 554 | - | expression tag |
Ser 555 | - | expression tag |
Glu 556 | - | expression tag |
Lys 557 | - | expression tag |
Met 558 | - | expression tag |
Lys 559 | - | expression tag |
Gly 560 | - | expression tag |
Met 561 | - | expression tag |
Lys 562 | - | expression tag |
Glu 563 | - | expression tag |
Leu 564 | - | expression tag |
Leu 565 | - | expression tag |
Val 566 | - | expression tag |
Ala 567 | - | expression tag |
Thr 568 | - | expression tag |
Lys 569 | - | expression tag |
Ile 570 | - | expression tag |
Asn 571 | - | expression tag |
Ser 572 | - | expression tag |
Ser 573 | - | expression tag |
Ala 574 | - | expression tag |
Ile 575 | - | expression tag |
Lys 576 | - | expression tag |
Leu 577 | - | expression tag |
Gln 578 | - | expression tag |
Leu 579 | - | expression tag |
Thr 580 | - | expression tag |
Ala 581 | - | expression tag |
Gln 582 | - | expression tag |
Ser 583 | - | expression tag |
Gln 584 | - | expression tag |
Val 585 | - | expression tag |
Gln 586 | - | expression tag |
Met 587 | - | expression tag |
Lys 588 | - | expression tag |
Lys 589 | - | expression tag |
Gln 590 | - | expression tag |
Lys 591 | - | expression tag |
Val 592 | - | expression tag |
Ser 593 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 56626.5 | |
Non-Polymers* | Number of molecules | 3 |
Total formula weight | 830.9 | |
All* | Total formula weight | 57457.4 |