4RT7
Crystal Structure of FLT3 with a small molecule inhibitor
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Receptor-type tyrosine-protein kinase FLT3 | polymer | 415 | 48200.3 | 1 | UniProt (P36888) Pfam (PF07714) In PDB | Homo sapiens (human) | FL cytokine receptor, Fetal liver kinase-2, FLK-2, Fms-like tyrosine kinase 3, FLT-3, Stem cell tyrosine kinase 1, STK-1 |
2 | A | 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-{7-[2-(morpholin-4-yl)ethoxy]imidazo[2,1-b][1,3]benzothiazol-2-yl}phenyl)urea | non-polymer | 560.7 | 1 | Chemie (P30) | |||
3 | water | water | 18.0 | 1 | Chemie (HOH) |
Sequence modifications
A: 564 - 958 (UniProt: P36888)
PDB | External Database | Details |
---|---|---|
Met 544 | - | EXPRESSION TAG |
Ser 545 | - | EXPRESSION TAG |
Tyr 546 | - | EXPRESSION TAG |
Tyr 547 | - | EXPRESSION TAG |
His 548 | - | EXPRESSION TAG |
His 549 | - | EXPRESSION TAG |
His 550 | - | EXPRESSION TAG |
His 551 | - | EXPRESSION TAG |
His 552 | - | EXPRESSION TAG |
His 553 | - | EXPRESSION TAG |
Ser 554 | - | EXPRESSION TAG |
Ser 555 | - | EXPRESSION TAG |
Gly 556 | - | EXPRESSION TAG |
Glu 557 | - | EXPRESSION TAG |
Asn 558 | - | EXPRESSION TAG |
Leu 559 | - | EXPRESSION TAG |
Tyr 560 | - | EXPRESSION TAG |
Phe 561 | - | EXPRESSION TAG |
Gln 562 | - | EXPRESSION TAG |
Gly 563 | - | EXPRESSION TAG |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 48200.3 | |
Non-Polymers* | Number of molecules | 1 |
Total formula weight | 560.7 | |
All* | Total formula weight | 48761.0 |