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7VV4

Cryo-EM structure of pseudoallergen receptor MRGPRX2 complex with linear cortistatin-14, local

Functional Information from GO Data
ChainGOidnamespacecontents
L0005179molecular_functionhormone activity
L0005576cellular_componentextracellular region
R0004930molecular_functionG protein-coupled receptor activity
R0005886cellular_componentplasma membrane
R0007186biological_processG protein-coupled receptor signaling pathway
R0016020cellular_componentmembrane
R0019233biological_processsensory perception of pain
R0030431biological_processsleep
R0032467biological_processpositive regulation of cytokinesis
R0042923molecular_functionneuropeptide binding
R0043303biological_processmast cell degranulation
R0045576biological_processmast cell activation
R1990595molecular_functionmast cell secretagogue receptor activity
Functional Information from PROSITE/UniProt
site_idPS00237
Number of Residues17
DetailsG_PROTEIN_RECEP_F1_1 G-protein coupled receptors family 1 signature. AGLsMLSTVSTERCLsV
ChainResidueDetails
RALA115-VAL131

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues75
DetailsTOPO_DOM: Extracellular => ECO:0000255
ChainResidueDetails
RMET1-PRO33
RASN85-SER96
RLYS166-ASP184
RTRP250-SER264

site_idSWS_FT_FI2
Number of Residues20
DetailsTRANSMEM: Helical; Name=1 => ECO:0000255
ChainResidueDetails
RVAL34-LEU54

site_idSWS_FT_FI3
Number of Residues100
DetailsTOPO_DOM: Cytoplasmic => ECO:0000255
ChainResidueDetails
RLEU55-ALA63
RSER118-HIS144
RLEU206-THR228
RARG286-VAL330

site_idSWS_FT_FI4
Number of Residues20
DetailsTRANSMEM: Helical; Name=2 => ECO:0000255
ChainResidueDetails
RPHE64-ILE84

site_idSWS_FT_FI5
Number of Residues20
DetailsTRANSMEM: Helical; Name=3 => ECO:0000255
ChainResidueDetails
RILE97-LEU117

site_idSWS_FT_FI6
Number of Residues20
DetailsTRANSMEM: Helical; Name=4 => ECO:0000255
ChainResidueDetails
RLEU145-GLY165

site_idSWS_FT_FI7
Number of Residues20
DetailsTRANSMEM: Helical; Name=5 => ECO:0000255
ChainResidueDetails
RPHE185-LEU205

site_idSWS_FT_FI8
Number of Residues20
DetailsTRANSMEM: Helical; Name=6 => ECO:0000255
ChainResidueDetails
RVAL229-ILE249

site_idSWS_FT_FI9
Number of Residues20
DetailsTRANSMEM: Helical; Name=7 => ECO:0000255
ChainResidueDetails
RVAL265-PHE285

221371

PDB entries from 2024-06-19

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