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7LDX

SARS-CoV-2 Main protease immature form - F2X Entry Library E06 fragment

Replaces:  7KW5
Functional Information from GO Data
ChainGOidnamespacecontents
A0008233molecular_functionpeptidase activity
A0019082biological_processviral protein processing
B0008233molecular_functionpeptidase activity
B0019082biological_processviral protein processing
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue PEG A 501
ChainResidue
AHOH616
BGLY79
BSER81
BLYS90

site_idAC2
Number of Residues3
Detailsbinding site for residue PEG A 502
ChainResidue
AGLN19
ALEU67
AASN119

site_idAC3
Number of Residues3
Detailsbinding site for residue PEG A 503
ChainResidue
BARG4
AGLU290
BPHE3

site_idAC4
Number of Residues9
Detailsbinding site for residue DMS A 504
ChainResidue
ALYS5
AALA7
AGLN127
AHOH657
BLYS5
BMET6
BALA7
BTYR126
BGLN127

site_idAC5
Number of Residues1
Detailsbinding site for residue DMS A 505
ChainResidue
AASN84

site_idAC6
Number of Residues2
Detailsbinding site for residue DMS A 506
ChainResidue
AGLN19
AGLY71

site_idAC7
Number of Residues2
Detailsbinding site for residue DMS A 507
ChainResidue
ALEU271
AGLY275

site_idAC8
Number of Residues3
Detailsbinding site for residue DMS A 508
ChainResidue
AMET6
APHE8
AHOH656

site_idAC9
Number of Residues7
Detailsbinding site for residue R9V A 509
ChainResidue
APRO132
AASN133
ATHR196
AMET235
ATYR239
AGLU240
APRO241

site_idAD1
Number of Residues6
Detailsbinding site for residue DMS B 401
ChainResidue
ASER123
BMET6
BPHE8
BGLN127
BASP295
BARG298

site_idAD2
Number of Residues5
Detailsbinding site for residue R9V B 402
ChainResidue
BPRO132
BASN133
BTHR196
BTHR198
BGLU240

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE: For 3CL-PRO activity => ECO:0000255|PROSITE-ProRule:PRU00772, ECO:0000305|PubMed:32198291
ChainResidueDetails
BHIS41
AHIS41

site_idSWS_FT_FI2
Number of Residues2
DetailsACT_SITE: Nucleophile; for 3CL-PRO activity => ECO:0000255|PROSITE-ProRule:PRU00772, ECO:0000269|PubMed:32198291
ChainResidueDetails
BCYS145
ACYS145

site_idSWS_FT_FI3
Number of Residues2
DetailsSITE: Cleavage; by 3CL-PRO => ECO:0000250|UniProtKB:P0C6V3
ChainResidueDetails
BGLN306
AGLN306

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PDB entries from 2024-06-12

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