7BJU
Crystal structure of the ligand-binding domains of the heterodimer EcR/USP bound to the synthetic agonist BYI08346
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0003677 | molecular_function | DNA binding |
A | 0003707 | molecular_function | nuclear steroid receptor activity |
A | 0005634 | cellular_component | nucleus |
A | 0006355 | biological_process | regulation of DNA-templated transcription |
A | 0008270 | molecular_function | zinc ion binding |
D | 0003677 | molecular_function | DNA binding |
D | 0004879 | molecular_function | nuclear receptor activity |
D | 0005634 | cellular_component | nucleus |
D | 0006355 | biological_process | regulation of DNA-templated transcription |
D | 0035076 | biological_process | ecdysone receptor-mediated signaling pathway |
D | 0035100 | molecular_function | ecdysone binding |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 11 |
Details | binding site for residue EPH A 501 |
Chain | Residue |
A | LEU230 |
A | LEU435 |
A | PHE438 |
A | PRO239 |
A | PHE242 |
A | LEU249 |
A | GLY328 |
A | SER335 |
A | GLN338 |
A | ALA339 |
A | HIS434 |
site_id | AC2 |
Number of Residues | 2 |
Details | binding site for residue PEG D 601 |
Chain | Residue |
A | LYS355 |
D | ASP448 |
site_id | AC3 |
Number of Residues | 15 |
Details | binding site for residue 834 D 602 |
Chain | Residue |
D | THR343 |
D | MET380 |
D | MET381 |
D | VAL384 |
D | TYR403 |
D | TYR408 |
D | VAL416 |
D | ASP419 |
D | LEU420 |
D | GLN503 |
D | ASN504 |
D | MET507 |
D | CYS508 |
D | LEU522 |
D | TRP526 |
site_id | AC4 |
Number of Residues | 6 |
Details | binding site for residue PE8 D 603 |
Chain | Residue |
D | SER296 |
D | SER296 |
D | ALA299 |
D | ARG300 |
D | TYR303 |
D | TYR303 |
site_id | AC5 |
Number of Residues | 2 |
Details | binding site for residue PGE D 604 |
Chain | Residue |
D | LYS362 |
D | TYR464 |
site_id | AC6 |
Number of Residues | 2 |
Details | binding site for residue MG D 605 |
Chain | Residue |
D | PHE353 |
D | GLY356 |