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7AXC

Crystal structure of the hPXR-LBD in complex with ferutinine

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue 27H A 501
ChainResidue
AMET243
ASER247
AGLN285
APHE288
ATRP299
AGLU321
AMET323
AHIS407

site_idAC2
Number of Residues6
Detailsbinding site for residue GOL A 502
ChainResidue
ALYS392
AALA395
AMET396
AHOH627
AHOH650
AMET159

site_idAC3
Number of Residues2
Detailsbinding site for residue IPA A 503
ChainResidue
AASN171
APHE172

site_idAC4
Number of Residues1
Detailsbinding site for residue IPA A 504
ChainResidue
ALYS160

site_idAC5
Number of Residues4
Detailsbinding site for residue IPA A 505
ChainResidue
ATHR290
AGLU337
AHOH620
AHOH629

site_idAC6
Number of Residues2
Detailsbinding site for residue IPA A 506
ChainResidue
ALEU276
AGLU427

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
ChainResidueDetails
AHIS407
ASER247
AGLN285

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PDB entries from 2024-06-12

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