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6YWZ

Crystal structure of SHANK1 PDZ in complex with a peptide-small molecule hybrid

Functional Information from PDB Data
site_idAC1
Number of Residues1
Detailsbinding site for residue PEG B 801
ChainResidue
BARG804

site_idAC2
Number of Residues5
Detailsbinding site for residue ARG B 804
ChainResidue
BVAL677
BASP706
BPEG801
BTHR803
BLEU805

site_idAC3
Number of Residues7
Detailsbinding site for residue LEU B 805
ChainResidue
BPHE676
BILE742
BTHR803
BARG804
BGLY673
BPHE674
BGLY675

site_idAC4
Number of Residues4
Detailsbinding site for residue ARG A 803
ChainResidue
APHE676
AASP706
ATHR802
ALEU804

site_idAC5
Number of Residues6
Detailsbinding site for residue LEU A 804
ChainResidue
AGLY673
APHE674
AGLY675
APHE676
AILE742
AARG803

site_idAC6
Number of Residues8
Detailsbinding site for Di-peptide PWN A 801 and THR A 802
ChainResidue
AVAL677
ALEU678
AARG679
AGLY680
AALA681
AGLN700
AHIS735
AARG803

site_idAC7
Number of Residues12
Detailsbinding site for Di-peptide PWN B 802 and THR B 803
ChainResidue
BVAL677
BLEU678
BARG679
BGLY680
BLYS682
BALA683
BHIS735
BARG743
BARG804
BLEU805
BHOH902
BHOH914

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0000250|UniProtKB:D3YZU1
ChainResidueDetails
ASER671
BSER671

219869

PDB entries from 2024-05-15

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