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6VPF

Estrogen Receptor Alpha Ligand Binding Domain in Complex with the Selective Estrogen Receptor Modulator Clomiphene

Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue 53Q B 601
ChainResidue
BMET343
BVAL533
BLEU346
BTHR347
BALA350
BASP351
BTRP383
BMET421
BILE424
BGLY521

site_idAC2
Number of Residues14
Detailsbinding site for residue 53Q A 601
ChainResidue
AMET343
ALEU346
ATHR347
AALA350
AASP351
AGLU353
ATRP383
ALEU387
AILE424
AGLY521
AHIS524
ALEU525
AASN532
AVAL533

site_idAC3
Number of Residues13
Detailsbinding site for residue 53Q C 601
ChainResidue
CMET343
CLEU346
CTHR347
CALA350
CASP351
CGLU353
CTRP383
CMET421
CGLY521
CHIS524
CLEU525
CASN532
CVAL533

site_idAC4
Number of Residues14
Detailsbinding site for residue 53Q D 601
ChainResidue
DMET343
DLEU346
DTHR347
DALA350
DASP351
DGLU353
DTRP383
DILE424
DGLY521
DHIS524
DLEU525
DASN532
DVAL533
DPRO535

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsMOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106
ChainResidueDetails
BTYR537
ATYR537
CTYR537
DTYR537

site_idSWS_FT_FI2
Number of Residues4
DetailsLIPID: S-palmitoyl cysteine => ECO:0000250
ChainResidueDetails
BCYS447
ACYS447
CCYS447
DCYS447

220113

PDB entries from 2024-05-22

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