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5V7T

crystal structure of PARP14 bound to N-{4-[4-(diphenylmethoxy)piperidin-1-yl]butyl}[1,2,4]triazolo[4,3-b]pyridazin-6-amine inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue 91V A 1801
ChainResidue
AHIS1601
AHIS1672
AHOH1928
AGLY1602
ALYS1630
ATYR1633
AASN1639
ATYR1640
ASER1641
ATYR1646
ATYR1646

219869

PDB entries from 2024-05-15

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