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5NFT

Glucocorticoid Receptor in complex with AZD5423

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue EDO A 801
ChainResidue
APRO541
AALA574
ATRP577
ALYS667
AHOH925
AHOH959

site_idAC2
Number of Residues1
Detailsbinding site for residue EDO A 802
ChainResidue
AHIS645

site_idAC3
Number of Residues2
Detailsbinding site for residue EDO A 803
ChainResidue
APRO750
AGLU751

site_idAC4
Number of Residues16
Detailsbinding site for residue 8W8 A 804
ChainResidue
AMET560
ALEU563
AASN564
ALEU566
AGLY567
AGLN570
AMET604
AALA607
ALEU608
AARG611
APHE623
AGLN642
ATYR735
ACYS736
ATHR739
APHE749

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO) => ECO:0000269|PubMed:12144530
ChainResidueDetails
ALYS703

219140

PDB entries from 2024-05-01

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