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5M6H

Small Molecule inhibitors of IAP

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 401
ChainResidue
ACYS300
ACYS303
AHIS320
ACYS327

site_idAC2
Number of Residues6
Detailsbinding site for residue NA A 402
ChainResidue
AHOH555
APHE272
APHE272
AHOH538
AHOH538
AHOH555

site_idAC3
Number of Residues12
Detailsbinding site for residue 7J6 A 403
ChainResidue
ALEU292
AVAL298
AGLY306
ALEU307
ATHR308
AASP309
ATRP310
ALYS311
AGLU314
AGLN319
ATRP323
ATYR324

Functional Information from PROSITE/UniProt
site_idPS01282
Number of Residues66
DetailsBIR_REPEAT_1 BIR repeat. YeaRiftfgt.Wiysvnkeqlar...AGFyAlgegDkvkCfhCgggltdWkpsedpweqHakwyPgCkyL
ChainResidueDetails
ATYR265-LEU330

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00029
ChainResidueDetails
ACYS300
ACYS303
AHIS320
ACYS327

site_idSWS_FT_FI2
Number of Residues3
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:12747801
ChainResidueDetails
ALYS328
ALYS322

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PDB entries from 2024-06-12

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