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4ZT5

Trypanosoma brucei methionyl-tRNA synthetase in complex with inhibitor (2S)-N-(3,5-dichlorobenzyl)-N'-(1H-imidazo[4,5-b]pyridin-2-yl)-2-methylpropane-1,3-diamine (Chem 1655)

Functional Information from GO Data
ChainGOidnamespacecontents
A0000166molecular_functionnucleotide binding
A0004812molecular_functionaminoacyl-tRNA ligase activity
A0004825molecular_functionmethionine-tRNA ligase activity
A0005524molecular_functionATP binding
A0006418biological_processtRNA aminoacylation for protein translation
A0006431biological_processmethionyl-tRNA aminoacylation
B0000166molecular_functionnucleotide binding
B0004812molecular_functionaminoacyl-tRNA ligase activity
B0004825molecular_functionmethionine-tRNA ligase activity
B0005524molecular_functionATP binding
B0006418biological_processtRNA aminoacylation for protein translation
B0006431biological_processmethionyl-tRNA aminoacylation
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue MET A 801
ChainResidue
AILE248
AHOH922
ATYR250
AASP287
ATRP474
AALA477
ATYR481
AILE519
AHIS523
ALYS550

site_idAC2
Number of Residues2
Detailsbinding site for residue GOL A 802
ChainResidue
AARG583
AARG601

site_idAC3
Number of Residues4
Detailsbinding site for residue DMS A 803
ChainResidue
ALYS521
AILE525
ADMS804
ADMS806

site_idAC4
Number of Residues5
Detailsbinding site for residue DMS A 804
ChainResidue
ALYS517
AASP518
ALEU520
ALYS521
ADMS803

site_idAC5
Number of Residues3
Detailsbinding site for residue DMS A 805
ChainResidue
ATRP345
AGLU349
APRO464

site_idAC6
Number of Residues2
Detailsbinding site for residue DMS A 806
ChainResidue
ALEU444
ADMS803

site_idAC7
Number of Residues3
Detailsbinding site for residue GOL B 801
ChainResidue
BARG583
BARG601
BHOH954

site_idAC8
Number of Residues6
Detailsbinding site for residue GOL B 802
ChainResidue
BGLU239
BARG279
BLYS442
BGLY443
BPRO445
BGLU506

site_idAC9
Number of Residues4
Detailsbinding site for residue DMS B 803
ChainResidue
BPHE319
BTYR324
BILE326
BHOH1072

site_idAD1
Number of Residues4
Detailsbinding site for residue DMS B 804
ChainResidue
BGLY573
BTYR574
BASP575
BHOH948

site_idAD2
Number of Residues4
Detailsbinding site for residue SO4 B 805
ChainResidue
BARG271
BVAL275
BSER714
BPRO718

site_idAD3
Number of Residues14
Detailsbinding site for residue 4RN B 806
ChainResidue
BILE248
BTYR250
BASP287
BHIS289
BGLY290
BVAL471
BVAL473
BTRP474
BASP476
BTYR481
BILE519
BHOH918
BHOH922
BHOH931

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PDB entries from 2024-06-12

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