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4YLU

X-ray structure of MERS-CoV nsp5 protease bound with a non-covalent inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0008233molecular_functionpeptidase activity
A0019082biological_processviral protein processing
B0008233molecular_functionpeptidase activity
B0019082biological_processviral protein processing
C0008233molecular_functionpeptidase activity
C0019082biological_processviral protein processing
D0008233molecular_functionpeptidase activity
D0019082biological_processviral protein processing
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue R30 A 401
ChainResidue
AHIS41
AGLN192
AHOH547
BSER1
ALEU49
APHE143
ACYS148
AHIS166
AMET168
AGLU169
AASP190
ALYS191

site_idAC2
Number of Residues2
Detailsbinding site for residue ACT A 402
ChainResidue
ATHR108
AASP181

site_idAC3
Number of Residues1
Detailsbinding site for residue ACT A 403
ChainResidue
AASP200

site_idAC4
Number of Residues12
Detailsbinding site for residue R30 B 401
ChainResidue
AHIS64
BMET25
BHIS41
BLEU49
BPHE143
BCYS148
BHIS166
BMET168
BGLU169
BASP190
BLYS191
BHOH674

site_idAC5
Number of Residues2
Detailsbinding site for residue ACT B 402
ChainResidue
BASP200
BHOH613

site_idAC6
Number of Residues12
Detailsbinding site for residue R30 C 401
ChainResidue
CMET25
CLEU49
CPHE143
CLEU144
CCYS148
CHIS166
CMET168
CGLU169
CASP190
CLYS191
CGLN192
DSER1

site_idAC7
Number of Residues1
Detailsbinding site for residue ACT C 402
ChainResidue
CASP200

site_idAC8
Number of Residues16
Detailsbinding site for residue R30 D 401
ChainResidue
DMET25
DHIS41
DCYS44
DALA46
DTYR54
DPHE143
DLEU144
DCYS145
DCYS148
DHIS166
DMET168
DGLU169
DASP190
DLYS191
DGLN192
DHOH540

site_idAC9
Number of Residues1
Detailsbinding site for residue ACT D 402
ChainResidue
DASP200

221051

PDB entries from 2024-06-12

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