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4DO0

Crystal Structure of human PHF8 in complex with Daminozide

Functional Information from PDB Data
site_idAC1
Number of Residues11
DetailsBINDING SITE FOR RESIDUE DZA A 501
ChainResidue
AILE191
AHOH611
AHOH612
ATHR244
AHIS247
AASP249
ATYR257
ALYS264
AHIS319
AVAL321
AZN502

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE ZN A 502
ChainResidue
AHIS247
AASP249
AHIS319
ADZA501
AHOH612

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 503
ChainResidue
ATHR143
AVAL144
AARG145
ATYR179
ATYR180
ALYS261

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 504
ChainResidue
AHIS395
AHIS395
ALYS398
ALYS398

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 505
ChainResidue
AASP131
AGLY132
ALEU133
AGLY134
AMET135

site_idAC6
Number of Residues2
DetailsBINDING SITE FOR RESIDUE SO4 A 506
ChainResidue
AARG145
AHIS149

site_idAC7
Number of Residues2
DetailsBINDING SITE FOR RESIDUE SO4 A 507
ChainResidue
ALYS208
AARG211

site_idAC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 508
ChainResidue
ATHR272
AASN273
AALA390
ASER391
ATYR392

site_idAC9
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 509
ChainResidue
AASP100
AGLU101
ALYS105
APRO106
APHE115

site_idBC1
Number of Residues1
DetailsBINDING SITE FOR RESIDUE ACT A 510
ChainResidue
AARG360

site_idBC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 511
ChainResidue
ASER141
AHIS149
AARG199

site_idBC3
Number of Residues2
DetailsBINDING SITE FOR RESIDUE EDO A 512
ChainResidue
ALYS302
ASER304

site_idBC4
Number of Residues2
DetailsBINDING SITE FOR RESIDUE ACT A 513
ChainResidue
AGLN110
ALYS299

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBINDING:
ChainResidueDetails
ATHR244
ALYS264

site_idSWS_FT_FI2
Number of Residues3
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00538, ECO:0000269|PubMed:20023638, ECO:0000269|PubMed:20101266
ChainResidueDetails
AHIS319
AHIS247
AASP249

site_idSWS_FT_FI3
Number of Residues1
DetailsMOD_RES: Phosphoserine; by CDK1 => ECO:0000269|PubMed:20622854, ECO:0007744|PubMed:23186163
ChainResidueDetails
ASER84

220472

PDB entries from 2024-05-29

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