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4BE2

PFV intasome with inhibitor XZ-259

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
B0003676molecular_functionnucleic acid binding
B0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 393
ChainResidue
AHIS62
AHIS66
ACYS96
ACYS99

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 B 1300
ChainResidue
BARG222
BSER258
BPRO259
BVAL260

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 1376
ChainResidue
ALYS339
AHIS357
AHOH2198
AHIS338

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE GOL A 1377
ChainResidue
ASER162
ATHR163
ASER164
AHOH2207

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE GOL A 1378
ChainResidue
APRO135
ASER136
AGLN137
ALYS241

site_idAC6
Number of Residues4
DetailsBINDING SITE FOR RESIDUE GOL B 1301
ChainResidue
BTYR263
BGLN267
BGLY271
BASP273

site_idAC7
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL A 1379
ChainResidue
AGLN60
ALEU79
ATYR80
APRO277
APHE278

site_idAC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE MG A 1380
ChainResidue
AASP128
AASP185
AHOH2069
AHOH2070
DXZ21018

site_idAC9
Number of Residues5
DetailsBINDING SITE FOR RESIDUE MG A 1381
ChainResidue
AASP128
AGLU221
AASN224
AHOH2071
DXZ21018

site_idBC1
Number of Residues15
DetailsBINDING SITE FOR RESIDUE XZ2 D 1018
ChainResidue
AASP128
AASP185
ATYR212
APRO214
AGLN215
AGLU221
AMG1380
AMG1381
ASO41382
AHOH2069
AHOH2070
AHOH2071
CDG4
DDC16
DDA17

site_idBC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE MG B 1302
ChainResidue
BASP128
BASP185
BHOH2012
BHOH2013
BHOH2031
CDA19

site_idBC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 1382
ChainResidue
AASP185
AGLN186
AGLY187
APRO211
ATYR212
DXZ21018

site_idBC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE GOL A 1383
ChainResidue
APRO115
AASP116
CDT3

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250
ChainResidueDetails
AASP123
AASP185
BASP123
BASP185

221051

PDB entries from 2024-06-12

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