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3PWW

Endothiapepsin in complex with saquinavir

Functional Information from GO Data
ChainGOidnamespacecontents
A0004190molecular_functionaspartic-type endopeptidase activity
A0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues22
DetailsBINDING SITE FOR RESIDUE ROC A 1001
ChainResidue
AASP15
APHE194
AILE217
AASP219
AGLY221
ATHR222
ATHR223
ATYR226
AILE304
AHOH392
AHOH503
AASP33
AHOH551
AHOH641
AHOH721
AASP35
AGLY37
ASER78
ATYR79
AGLY80
AASP81
APHE116

site_idAC2
Number of Residues9
DetailsBINDING SITE FOR RESIDUE GOL A 3002
ChainResidue
AVAL272
APRO274
ATYR277
AALA312
ASER329
ALYS330
AHOH379
AHOH445
AHOH598

Functional Information from PROSITE/UniProt
site_idPS00141
Number of Residues12
DetailsASP_PROTEASE Eukaryotic and viral aspartyl proteases active site. LDFDTGSSDLWV
ChainResidueDetails
ALEU32-VAL43
AGLY216-LEU227

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE:
ChainResidueDetails
AASP35
ASER199

220472

PDB entries from 2024-05-29

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