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3PB9

Crystal structure of the catalytic domain of human Golgi-resident glutaminyl cyclase in complex with 1-benzylimidazole

Functional Information from GO Data
ChainGOidnamespacecontents
X0016603molecular_functionglutaminyl-peptide cyclotransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues9
DetailsBINDING SITE FOR RESIDUE 1BN X 390
ChainResidue
XASP186
XGLU225
XGLU226
XTRP231
XASP269
XGLU325
XTRP350
XHIS351
XZN400

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN X 400
ChainResidue
XASP186
XGLU226
XHIS351
X1BN390

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE: Proton acceptor => ECO:0000250|UniProtKB:Q16769
ChainResidueDetails
XGLU225
XASP269

site_idSWS_FT_FI2
Number of Residues3
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:Q16769
ChainResidueDetails
XASP186
XGLU226
XHIS351

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PDB entries from 2024-04-24

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